Studies on 1,4-benzothiazines. IV. Reactions of 2-acyl-4H-1,4-benzothiazines with hydroxylamine, hydrazine, guanidine and acetamidine.
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2-Acyl-4-methyl-4H-1, 4-benzothiazines (1a, b) reacted with hydroxylamine to give dihydroisoxazolo [4, 5-b] [1, 4] benzothiazines (3a, b). However, the reaction of 1a with hydrazine did not give the dihydropyrazolo [4, 5-b] [1, 4] benzothiazine derivative corresponding to 3a, but gave its dehydro compound (6). On the other hand, in the reaction of 1b with hydrazine, formation of a pyrazole ring and opening of the thiazine ring occurred to afford a 4-(2-aminophenylthio) pyrazole derivative (7). Guanidine and acetamidine also reacted with 1a, b to give 5-[2-(N-methylamino) phenylthio] pyrimidines (10a-d).
収録刊行物
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- CHEMICAL & PHARMACEUTICAL BULLETIN
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CHEMICAL & PHARMACEUTICAL BULLETIN 32 (4), 1593-1596, 1984
公益社団法人 日本薬学会
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詳細情報 詳細情報について
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- CRID
- 1390001204167086976
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- NII論文ID
- 110003624941
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- NII書誌ID
- AA00602100
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- ISSN
- 13475223
- 00092363
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- 本文言語コード
- en
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- データソース種別
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- JaLC
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- CiNii Articles
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- 抄録ライセンスフラグ
- 使用不可