PAYNE REARRANGEMENT ROUTE TO THE OPTICALLY ACTIVE OXIRANE PRECURSOR FOR THE PREPARATION OF TRIAZOLE ANTIFUNGALS

Abstract

Optically active epoxide 1,an important intermediate for the preparation of antifungal triazole-amides 2,was synthesized starting from the (S)-lactic acid- derived ketone 9 and taking advantage of the Payne rearrangement of the epoxyalocohol 8.

Journal

Chemical & pharmaceutical bulletin   [List of Volumes]

Chemical & pharmaceutical bulletin 40(2), 562-564, 1992-02-25  [Table of Contents]

The Pharmaceutical Society of Japan

Cited by:  3

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Codes

  • NII Article ID (NAID) :
    110003629816
  • NII NACSIS-CAT ID (NCID) :
    AA00602100
  • Text Lang :
    ENG
  • Article Type :
    Journal Article
  • ISSN :
    00092363
  • Databases :
    CJPref  NII-ELS