Synthesis and Fungicidal Activities of Phenoxyphenyl Alkoxyiminoacetamide Derivatives

DOI NDL Digital Collections JASI Web Site Web Site 10 Citations 18 References

Bibliographic Information

Other Title
  • フェノキシフェニルアルコキシイミノアセトアミド誘導体の合成と殺菌活性
  • Synthesis and Fungicidal Activities of
  • Structure and Fungicidal Activities of New Alkoxyiminoacetamide Derivatives (Part 1)

Search this article

Abstract

A number of alkoxyiminophenylacetamide derivatives were synthesized and their fungicidal activities were examined. Studies of structure-activity relationships revealed strongest fungicidal activity when the alkoxyimino moiety and the acetamide moiety were each substituted with a methyl group. When the 2-position of the benzene ring on the phenylacetamide moiety was substituted with a phenoxy or phenoxymethyl group, good fungicidal activity was obtained. Introduction of other substituents on the benzene ring of the phenylacetamide moiety resulted in decrease of the fungicidal activity. However, introduction of some substituents on the benzene ring of the 2-phenoxy group increased the activity to some extent. Between the two oxime geometrical isomers, the activity of the E-form was much stronger than that of the Z-form. Consequently, (E)-2-methoxyimino-N-methyl-2-(2-phenoxyphenyl)acetamide was selected as a candidate fungicide for rice diseases.

Journal

Citations (10)*help

See more

References(18)*help

See more

Keywords

Details 詳細情報について

Report a problem

Back to top