Structure−Activity Relationship Studies of Salinosporamide A (NPI-0052), a Novel Marine Derived Proteasome Inhibitor

  • Venkat R. Macherla
    Nereus Pharmaceuticals, Inc., 10480 Wateridge Circle, San Diego, California 92121, and Center for Marine Biotechnology and Biomedicine, Scripps Institution of Oceanography, University of California, San Diego, La Jolla, California 92093
  • Scott S. Mitchell
    Nereus Pharmaceuticals, Inc., 10480 Wateridge Circle, San Diego, California 92121, and Center for Marine Biotechnology and Biomedicine, Scripps Institution of Oceanography, University of California, San Diego, La Jolla, California 92093
  • Rama Rao Manam
    Nereus Pharmaceuticals, Inc., 10480 Wateridge Circle, San Diego, California 92121, and Center for Marine Biotechnology and Biomedicine, Scripps Institution of Oceanography, University of California, San Diego, La Jolla, California 92093
  • Katherine A. Reed
    Nereus Pharmaceuticals, Inc., 10480 Wateridge Circle, San Diego, California 92121, and Center for Marine Biotechnology and Biomedicine, Scripps Institution of Oceanography, University of California, San Diego, La Jolla, California 92093
  • Ta-Hsiang Chao
    Nereus Pharmaceuticals, Inc., 10480 Wateridge Circle, San Diego, California 92121, and Center for Marine Biotechnology and Biomedicine, Scripps Institution of Oceanography, University of California, San Diego, La Jolla, California 92093
  • Benjamin Nicholson
    Nereus Pharmaceuticals, Inc., 10480 Wateridge Circle, San Diego, California 92121, and Center for Marine Biotechnology and Biomedicine, Scripps Institution of Oceanography, University of California, San Diego, La Jolla, California 92093
  • Gordafaried Deyanat-Yazdi
    Nereus Pharmaceuticals, Inc., 10480 Wateridge Circle, San Diego, California 92121, and Center for Marine Biotechnology and Biomedicine, Scripps Institution of Oceanography, University of California, San Diego, La Jolla, California 92093
  • Bao Mai
    Nereus Pharmaceuticals, Inc., 10480 Wateridge Circle, San Diego, California 92121, and Center for Marine Biotechnology and Biomedicine, Scripps Institution of Oceanography, University of California, San Diego, La Jolla, California 92093
  • Paul R. Jensen
    Nereus Pharmaceuticals, Inc., 10480 Wateridge Circle, San Diego, California 92121, and Center for Marine Biotechnology and Biomedicine, Scripps Institution of Oceanography, University of California, San Diego, La Jolla, California 92093
  • William F. Fenical
    Nereus Pharmaceuticals, Inc., 10480 Wateridge Circle, San Diego, California 92121, and Center for Marine Biotechnology and Biomedicine, Scripps Institution of Oceanography, University of California, San Diego, La Jolla, California 92093
  • Saskia T. C. Neuteboom
    Nereus Pharmaceuticals, Inc., 10480 Wateridge Circle, San Diego, California 92121, and Center for Marine Biotechnology and Biomedicine, Scripps Institution of Oceanography, University of California, San Diego, La Jolla, California 92093
  • Kin S. Lam
    Nereus Pharmaceuticals, Inc., 10480 Wateridge Circle, San Diego, California 92121, and Center for Marine Biotechnology and Biomedicine, Scripps Institution of Oceanography, University of California, San Diego, La Jolla, California 92093
  • Michael A. Palladino
    Nereus Pharmaceuticals, Inc., 10480 Wateridge Circle, San Diego, California 92121, and Center for Marine Biotechnology and Biomedicine, Scripps Institution of Oceanography, University of California, San Diego, La Jolla, California 92093
  • Barbara C. M. Potts
    Nereus Pharmaceuticals, Inc., 10480 Wateridge Circle, San Diego, California 92121, and Center for Marine Biotechnology and Biomedicine, Scripps Institution of Oceanography, University of California, San Diego, La Jolla, California 92093

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