From structure to clinical development : allosteric modulation of G protein-coupled receptors
Author(s)
Bibliographic Information
From structure to clinical development : allosteric modulation of G protein-coupled receptors
(Advances in pharmacology / edited by Silvio Garattini [and] Parkhurst A. Shore, v. 88)
Academic Press, 2020
- hbk.
Available at 3 libraries
  Aomori
  Iwate
  Miyagi
  Akita
  Yamagata
  Fukushima
  Ibaraki
  Tochigi
  Gunma
  Saitama
  Chiba
  Tokyo
  Kanagawa
  Niigata
  Toyama
  Ishikawa
  Fukui
  Yamanashi
  Nagano
  Gifu
  Shizuoka
  Aichi
  Mie
  Shiga
  Kyoto
  Osaka
  Hyogo
  Nara
  Wakayama
  Tottori
  Shimane
  Okayama
  Hiroshima
  Yamaguchi
  Tokushima
  Kagawa
  Ehime
  Kochi
  Fukuoka
  Saga
  Nagasaki
  Kumamoto
  Oita
  Miyazaki
  Kagoshima
  Okinawa
  Korea
  China
  Thailand
  United Kingdom
  Germany
  Switzerland
  France
  Belgium
  Netherlands
  Sweden
  Norway
  United States of America
Note
Serial editor: S.J. Enna
Managing editor: Lynn Lecount
Description and Table of Contents
Description
From Structure to Clinical Development: Allosteric Modulation of G Protein-Coupled Receptors, Volume 88, the latest release in the Advances in Pharmacology series, presents a variety of chapters from the best authors in the field. Chapters in this updated edition include Targeting muscarinic M1 receptor in neurodegeneration, Photo-switchable allosteric ligands, Computational approaches for the design of mGlu receptor allosteric modulators, Allosteric modulation of GLP-1 receptor in metabolic disorders, Group II mGluR roles in the nervous system and their roles in addiction, RAMPs as allosteric modulators of Class B GPCRs, Structure-based discovery and development of mGlu5 NAMs, and much more.
Table of Contents
The computational modeling of allosteric modulation of metabotropic glutamate receptors
Laura Perez-Benito, Claudia Llinas del Torrent, Leonardo Pardo and Gary Tresadern
Structure-based discovery and development of metabotropic glutamate receptor 5 negative allosteric modulators
Kirstie A. Bennett, John A. Christopher and Benjamin G. Tehan
The function and allosteric control of the human sweet taste receptor
Guy Servant, Terry Kenakin, Lan Zhang, Mark Williams and Nicole Servant
The different aspects of the GABAB receptor allosteric modulation
Julie Kniazeff
RAMPs as allosteric modulators of the calcitonin and calcitonin-like class B G protein-coupled receptors
Augen A. Pioszak and Debbie L. Hay
Strategies and considerations of G-protein-coupled receptor photopharmacology
Alice E. Berizzi and Cyril Goudet
Discovery and pharmacology of the covalent GLP-1 receptor (GLP-1R) allosteric modulator BETP. A novel tool to probe GLP-1R pharmacology
Francis S. Willard, Joseph D. Ho and Kyle W. Sloop
Allosteric modulation of metabotropic glutamate receptors in alcohol use disorder: Insights from preclinical investigations
Kari A. Johnson and David M. Lovinger
Allosteric modulation of muscarinic receptors in alcohol and substance use disorders
Leigh C. Walker and Andrew J. Lawrence
M1 muscarinic acetylcholine receptors: A therapeutic strategy for symptomatic and disease-modifying effects in Alzheimer's disease?
Miriam Scarpa, Sarah Hesse and Sophie J. Bradley
by "Nielsen BookData"