The ADME encyclopedia : a comprehensive guide on biopharmacy and pharmacokinetics
著者
書誌事項
The ADME encyclopedia : a comprehensive guide on biopharmacy and pharmacokinetics
Springer, 2022
- hbk.
大学図書館所蔵 全1件
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内容説明・目次
内容説明
The ADME Encyclopedia covers pharmacokinetic phenomena (Absorption, Distribution, Metabolism and Excretion processes) and their relationship with the design of pharmaceutical carriers and the success of drug therapies. It covers both basic and advanced knowledge, serving as introductory material for students of biomedical careers and also as reference, updated material for graduates and professionals working in any field related to pharmaceutical sciences (medicine, pharmaceutical technology, materials science, medicinal chemistry).
Structured as alphabetically ordered entries with cross-references, the Encyclopedia not only provides basic knowledge on ADME processes, but also detailed entries on some advanced subjects such as drug transporters, last generation pharmaceutical carriers, pharmacogenomics, personalized medicine, bioequivalence studies, biowaivers, biopharmaceuticals, gene delivery, pharmacometrics, pharmacokinetic drug interactions or in silico and in vitro assessment of ADME properties
目次
Drug dissolution and drug release
Mathematical models of drug dissolution and drug release
Diffusion layer model
Danckwert's model
Interfacial barrier model
First order model
Higuchi model
Korsmeyer-Peppas model
Hixson-Crowell model
Baker-Lonsdale model
Weibull model
In vitro dissolution testing
Modalities of dissolution tests
Biorelevant dissolution media
Drug absorption
Free diffusion
Facilitated diffusion
Active transport
Transcytosis
pH partition theory
pKa determination
Factors impacting drug absorption
Drug distribution
Factors impacting drug distribution
Real volume of distribution
Apparent volume of distribution
Drug binding to plasma proteins
Drug displacement
Non-linear binding to plasma proteins
Drug binding to tissue components
One-compartment pharmacokinetic model
Two-compartment pharmacokinetic model
Central nervous system bioavailability
Blood-brain barrier
log BB
Kpuu
Drug metabolism
Functionalization reactions
Synthetic reactions
Cytochrome P450
Phase III reactions
Factors impacting on drug metabolism
Genetic variants. Polymorphism
Age
Gender
Environmental factors: enzyme induction
Precision medicine
Pharmacogenomic DNA chips
Microsomes
Drug excretion
Biliary excretion
Enterohepatic recycling
Enterohepatic recycling and antibiotics
Renal excretion
Glomerular filtration
Tubular reabsorption
Tubular secretion
Clearance
Organ clearance
Routes of administration
Oral route
Migrating motor complex
Enteric coating tablets
Food-drug interactions
Gastric emptying
Gastroretentive drug delivery systems
Multiparticulate drug delivery systems
Gut microbiota
Lipinski rule of five
Permeation enhancers
Intestinal perfusion models
Bucal and sublingual route
Rectal route
Intravenous route
Intravenous bolus
Intravenous infusion
Technological considerations for intravenous administration
Intramuscular administration
Subcutaneous administration
Specialized parenteral routes
Pulmonary administration
Nasal administration
Transdermal administration
Permeation enhancers
Next generation drug delivery systems
Nanocarriers
Surface-to-volume ratio
Surface chemistry
Nanotoxicology
Drug release from nanocarriers
Passive targeting
Smart systems / stimuli-responsive systems
Active targeting
Mononuclear phagocyte system
Absorption and distribution of nanocarriers
Elimination of nanocarriers
PEGylationADME
Viral vectors
Pharmacogenomics
Enzyme polymorphism
Transporter polymorphism
Pharmacogenomics and pediatrics
Bioavailability and bioequivalence
Bioavailability
Systemic bioavailability
Generic drugs
Post-approval changes
Bioequivalence
Absolute bioavailability
Mass balance studies
Bioequivalence studies
Reference and test products
Biopharmaceutical Classification System
Biowaivers
BCS subclasses
Dissolution testing
Pharmacodynamic studies
Biopharmaceutical drug products
Absorption of protein drugs
Distribution of protein drugs
Elimination of protein drugs
ADME properties of insulins
ADME properties of heparins
ADME properties of gene-based biopharmaceuticals
Drug-drug and food-drug interactions
Plasma protein binding DDI
Membrane transport DDI
Metabolism DDI
FDI based on induction of gastrointestinal changes
In vitro and in silico ADME predictions
Polarized cell lines
Caco-2
MDCK
Solubility
Dissolution testing
QSPR/QSAR
Expert rules
Central Nervous System Multiparameter Optimization
Dynamic transit models
Sandwich-cultured hepatocytes
Single-cell expression systems
Membrane vesicles
Molecular dynamics simulations
Drug tansporters
ABC transporters
MDR1
MRPs
BCRP
Solute carriers
Organic anion transporters
Organic cation transporters
Peptide transporters
Non-linear pharmacokinetics
Linear pharmacokinetics
Positive deviations from linear behavior
Negative deviations from linear behavior
Time-dependent pharmacokinetics
Pharmacometrics and physiologic models
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